Catalog Number: |
D24056 |
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CAS No.: |
N.A. |
MDL: |
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Formula: |
C24H28D3F6N3O7S |
F.W.: |
622.59 |
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Purity: |
99% |
Package: |
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Unit: |
mg |
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B.P.: |
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Density: |
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Optical Rotation: |
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Refractive Index: |
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Category: |
Reference Standard |
Reference: |
Koh, Y., et al.: Antimicrob. Agents Chemother., 47, 3123 (2003); Arasteh, K., et al.: AIDS, 19, 943 (2005); Surleraux, D.L.N.G., et al.: J. Med. Chem., 48, 1813 (2005) |
Application: |
4-Amino-N-((2R,3R)-3-amino-2-hydroxy-4-phenylbutyl)-N-isobutylbenzenesulfonamide-d9 Bis(2,2,2-trifluoroacetate) is the labeled analogue of 4-Amino-N-((2R,3R)-3-amino-2-hydroxy-4-phenylbutyl)-N-isobutylbenzenesulfonamide Bis(2,2,2-trifluoroacetate) ; an intermediate in the synthesis of 1-epi-Darunavir, a stereoisomer to Darunavir, a second generation HIV-1-protease inhibitor; structurally similar to amprenavir. Antiviral. |
Category: |
Amines, Aromatics, Metabolites & Impurities, Pharmaceuticals, Intermediates & Fine Chemicals, Sulfur & Selenium Compounds |