EPZ011989 |
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| Synonyms: N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl((1r,4r)-4-((2-methoxyethyl)(methyl)amino)cyclohexyl)amino)-2-methyl-5-(3-morpholinoprop-1-ynyl)benzamide;N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl-[4-[2-methoxyethyl(methyl)amino]cyclohexyl]amino]-2-methyl-5-(3-morpholin-4-ylprop-1-ynyl)benzamide;EPZ-011989, EPZ 011989 | |
| Cat. No.: E98000 | CAS No.: 1598383-40-4 |
| MDL.: | Formula: C35H51N5O4 |
| F.W.604.82 | Purity: 99% |
| Storage: | |
| Size/Unit | Price | Qty | Availability | Price Total |
|---|---|---|---|---|
| 5mg | $299.00 | Enter qty and click checkbox |
 
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$299.00 |
| Catalog Number： | E98000 | CAS No.: | 1598383-40-4 | |
| MDL: | Formula: | C35H51N5O4 | ||
| F.W.: | 604.82 | Purity: | 99% | |
| Package: | Unit: | mg | ||
| Appearance: | M.P.: | |||
| B.P.: | Density: | |||
| Optical Rotation: | Refractive Index: | |||
| Solubility: | DMSO | Stability: | ||
| Storage: | Category: | Reference Standard | ||
| Reference: | John E. Campbell et. al., ACS Med. Chem. Lett., 2015, 6 (5), pp 491–495 | |||
| Application: | EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. | |||