| Catalog Number: |
S12070 |
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CAS No.: |
N.A |
| MDL: |
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Formula: |
C16¹³C3H25N3O3 |
| F.W.: |
346.4 |
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Purity: |
99% |
| Package: |
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Unit: |
mg |
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Density: |
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Refractive Index: |
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Category: |
Reference Standard |
| Reference: |
Feng, J., et al.: J. Med. Chem., 50, 2297 (2007); Rosenstock, J., et al.: Diabetes Obes. Metab., 10, 376 (2008); Thomas, L., et al.: J. Pharmacol. Exp. Ther., 325, 175 (2008) |
| Application: |
N-Formyl Saxagliptin-13C3 is the labeled analogue of N-Formyl Saxagliptin (F701070), an impurity of Saxagliptin , a potent and selective reversible inhibitor of dipeptidyl peptidase-4, which is being developed for the treatment of type 2 diabetes. It is absorbed rapidly after oral administration and has a pharmacokinetic profile compatible with once daily dosing. |
| Category: |
Amines, Chiral Reagents, Heterocycles, Impurities, Isotope Labelled Compounds, Pharmaceuticals, Intermediates & Fine Chemicals |