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Entospletinib (GS-9973)

Synonyms: 6-(1H-Indazol-6-yl)-N-[4-(4-morpholinyl)phenyl]-Imidazo[1,2-a]pyrazin-8-amine;
Cat. No.: E08600 CAS No.: 1229208-44-9
MDL.: Formula: C23H21N7O
F.W.411.46 Purity: 99%
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Catalog Number: E08600   CAS No.: 1229208-44-9
MDL: Formula: C23H21N7O
F.W.: 411.46 Purity: 99%
Package: Unit: mg
Appearance: M.P.:
B.P.: Density:
Optical Rotation: Refractive Index:
Solubility: Stability:
Storage: Category: Reference Standard
Reference: Currie, K.S., et. al.: J. Med. Chem., 57, 3856 (2014)
Application: GS 9973 is a selective and orally bioavailable inhibitor of spleen tyrosine kinase (Syk).
Category: Amines, Aromatics, Inhibitors, Pharmaceuticals, Intermediates & Fine Chemicals